missing translation for 'onlineSavingsMsg'
Learn More
  1. Home
  2. Products
  3. Chemicals
  4. Organic compounds
  5. Organoheterocyclic compounds
  6. Indoles and derivatives
  7. CI 988, Tocris Bioscience™

CI 988, Tocris Bioscience™

Product Code. 18063782
Click to view available options
Quantity:
10 mg
50 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Potent and selective CCK2 antagonist

Potent and selective CCK2 (CCK-B) receptor antagonist that displays ∽ 1600-fold selectivity over CCK1 receptors (IC50 values are 1.7 and 2717 nM for CCK2 and CCK1 respectively). Has negligible affinity at a range of other binding sites (IC50 > 10 μM). Exhibits anxiolytic activity following oral administration.

Chemical Identifiers

CAS 130332-27-3
Molecular Formula C35H42N4O6
Molecular Weight (g/mol) 614.743
InChI Key FVQSSYMRZKLFDR-ZABPBAJSSA-N
Synonym unii-2637pdx9si, 3-1r-2-2r-2-2-adamantyloxycarbonylamino-3-1h-indol-3-yl-2-methyl-propanoyl amino-1-phenyl-ethyl carbamoyl propanoic acid, 4-1r-2-2r-2-2-adamantyloxycarbonylamino-3-1h-indol-3-yl-2-methylpropanoyl amino-1-phenylethyl amino-4-oxobutanoic acid, 4-1r-2-2r-3-1h-indol-3-yl-2-methyl-1-oxo-2-tricyclo 3.3.1.13,7 dec-2-yloxy carbonyl amino propyl amino-1-phenylethyl amino-4-oxobutanoic acid, gtpl873, butanoic acid, 4-1r-2-2r-3-1h-indol-3-yl-2-methyl-1-oxo-2-tricyclo 3.3.1.1 3,7 dec-2-yloxy carbonyl amino propyl amino-1-phenylethyl amino-4-oxo, r-r*,r*-4-2-3-1h-indol-3-yl-2-methyl-1-oxo-2-tricyclo 3.3.1.13,7 dec-2-yloxy carbonyl amino propyl amino-1-phenylethyl amino-4-oxobutanoic acid, 3-1r-2-2r-2-1h-indol-3-ylmethyl-2-1r,3r,5r,7r-adamantan-2-yloxy carbonyl amino propanamido-1-phenylethyl carbamoyl propanoic acid, 3-1r-2-2r-2-adamantan-2-yloxy carbonyl amino-2-1h-indol-3-ylmethyl propanamido-1-phenylethyl carbamoyl propanoic acid, 4-r-2-r-2-adamantan-2-yloxy carbonyl amino-3-1h-indol-3-yl-2-methylpropanamido-1-phenylethyl amino-4-oxobutanoic acid
PubChem CID 108187
IUPAC Name 4-[[(1R)-2-[[(2R)-2-(2-adamantyloxycarbonylamino)-3-(1H-indol-3-yl)-2-methylpropanoyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid
SMILES CC(CC1=CNC2=CC=CC=C21)(C(=O)NCC(C3=CC=CC=C3)NC(=O)CCC(=O)O)NC(=O)OC4C5CC6CC(C5)CC4C6

Specifications

Quantity 10 mg
Formula Weight 614.73
Percent Purity >99%
Chemical Name or Material CI 988
Product Content Correction

Your input is important to us. Please complete this form to provide feedback related to the content on this product.

Product Title

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.

Thank You! Your feedback has been submitted. Fisher Scientific is always working to improve our content for you. We appreciate your feedback.